SCHEMBL28025012

SCHEMBL28025012

COC(=O)c1c(C(F)(F)F)[nH]c2c(C)cccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.49
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 1/20 0.40
RPA1 P27694 1/20 0.39
MCL1 Q07820 1/20 0.39
LMNA P02545 2/20 0.38
ATM Q13315 1/20 0.38
MAPK1 P28482 1/20 0.38
AHR P35869 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28025010 0.85 GAA (0.53) NR4A2CA12CA1CA2CA7
SCHEMBL28025015 0.85 NR4A2 (0.50) NR4A2CA12CA1CA2CA7
SCHEMBL28207493 0.84 RPA1 (0.48) KMT2AMAPTKDM4EMEN1GAA
SCHEMBL28206982 0.84 PBRM1 (0.42) NR4A2CA12CA1CA2CA7
SCHEMBL28025006 0.83 KDM4E (0.49) NR4A2CA12CA1CA2CA7
SCHEMBL28024562 0.82 LMNA (0.52) MAPTKDM4EGAALMNAALDH1A1
SCHEMBL28024555 0.81 ALDH1A1 (0.37) NR4A2KMT2AMAPTKDM4EMEN1
SCHEMBL20867843 0.78 NR4A2 (0.63) NR4A2KMT2AMAPTKDM4EMEN1
SCHEMBL31312746 0.76 NR4A2 (0.50) NR4A2MAPTGAARPA1MCL1
SCHEMBL28024557 0.72 NR4A2 (0.49) NR4A2KMT2AMAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646327-A 2-perfluoroalkyl indole derivative and synthesis method thereof 上海大学 2016-06-08 CN disclosed
CN-104892485-A 2-perfluoroalkyl indole derivative and synthesis method thereof UNIV SHANGHAI 2015-09-09 CN disclosed