SCHEMBL28025571

SCHEMBL28025571

Cc1c(CC(=O)O)ccc2[nH]ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
TSHR P16473 2/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
GLA P06280 1/20 0.46
CYP2C9 P11712 1/20 0.46
NFKB1 P19838 1/20 0.46
PMP22 Q01453 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 6/20 0.46
P2RX7 Q99572 2/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
MAPT P10636 6/20 0.39
MEN1 O00255 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13820047 0.80 P2RX7 (0.40) P2RX7MTNR1AMTNR1B
SCHEMBL5376011 0.80 KDM4E (0.52) ALDH1A1TSHRHPGDLMNAGLA
SCHEMBL21617923 0.78 SMN1; SMN2 (0.51) GLAKDM4EMAPTMEN1KMT2A
SCHEMBL28947821 0.77 CYP1A2 (0.44) ALDH1A1TSHRHPGDLMNAGLA
SCHEMBL30009880 0.76 GRIN2D (0.54) ALDH1A1TSHRHPGDLMNAGLA
SCHEMBL4309213 0.76 GRIN2D (0.54) ALDH1A1TSHRHPGDLMNAGLA
SCHEMBL27973166 0.75 MPL (0.44) ALDH1A1TSHRHPGDLMNAGLA
SCHEMBL11741944 0.75 SRC (0.52) GLAKDM4EGRIN2DGRIN3BGRIN1
SCHEMBL29322645 0.75 HTR2B (0.40) TSHRNFKB1NPSR1P2RX7MAPT
SCHEMBL28025050 0.75 P2RX7 (0.46) ALDH1A1TSHRHPGDLMNAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854087-A As P2X7Indole carboxamide derivatives of receptor antagonists ACTELION PHARMACEUTICALS LTD 2015-08-19 CN disclosed
CN-104812749-A Iindole carboxamide derivatives as p2x7 receptor antagonists ACTELION PHARMACEUTICALS LTD 2015-07-29 CN disclosed