SCHEMBL28026053

SCHEMBL28026053

COC(=O)C(C)(CCC=O)S(C)(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.34
SLC6A2 P23975 1/20 0.30
MMP12 P39900 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17830429 0.83 PKM (0.38)
SCHEMBL12985153 0.83 PKM (0.38)
SCHEMBL17818301 0.79 ACLY (0.37) SLC6A2MMP12MMP13
SCHEMBL17818345 0.79 ACLY (0.37) SLC6A2MMP12MMP13
SCHEMBL19989708 0.79 DGAT1 (0.33) DGAT1SLC6A2MMP12MMP13
SCHEMBL20001472 0.77
SCHEMBL20001509 0.76 PAOX (0.33)
SCHEMBL28140457 0.75 DGAT1 (0.35) DGAT1SLC6A2MMP12MMP13
SCHEMBL27359921 0.75 DGAT1 (0.35) DGAT1
SCHEMBL3183165 0.75 DGAT1 (0.35) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311828-A Crystalline forms of (R) -4- (5- (cyclopropylethynyl) isoxazol-3-yl) -N-hydroxy-2-methyl-2- (methylsulfonyl) butanamide as antibacterial agents 诺华股份有限公司 2019-02-05 CN disclosed
CN-107001295-A Isoxazole hydroxamic acid compounds as lpxc inhibitors 诺华股份有限公司 2017-08-01 CN disclosed
CN-103717582-B As the different * oxazole derivatives of antiseptic-germicide PFIZER INC. (US) 2015-09-30 CN disclosed