SCHEMBL28026353

SCHEMBL28026353

CC(Oc1ccncc1Br)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.34
LATS1 O95835 1/20 0.33
LATS2 Q9NRM7 1/20 0.33
CA12 O43570 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
CA1 P00915 2/20 0.33
SLC6A9 P48067 2/20 0.32
GPR88 Q9GZN0 2/20 0.31
DHODH Q02127 4/20 0.31
CNR2 P34972 2/20 0.31
CA14 Q9ULX7 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP3A5 P20815 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
CHUK O15111 1/20 0.31
PRKD3 O94806 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15777428 1.00 RORC (0.34) RORCLATS1LATS2CA12CA2
SCHEMBL20481226 0.80 CA12 (0.37) CA12CA2CA9CA1CA14
SCHEMBL24200150 0.79 CA12 (0.36) CA12CA2CA9CA1CA14
SCHEMBL13724635 0.77 KDM4E (0.36) CA12CA2CA9CA1CA14
SCHEMBL15776169 0.77 CA12 (0.33) CA12CA2CA9CA1CA14
SCHEMBL527070 0.74 CA12 (0.33) CA12CA2CA9CA1CA14
SCHEMBL15475790 0.73 CA12 (0.33) CA12CA2CA9CA1CA14
SCHEMBL28715395 0.73 ALPL (0.39) CA12CA2CA9CA1CA14
SCHEMBL29421207 0.73 ALPL (0.39) CA12CA2CA9CA1CA14
SCHEMBL28026358 0.73 CNR2 (0.44) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837818-A Pyridine-2-amides useful as CB2 agonists HOFFMANN LA ROCHE 2015-08-12 CN disclosed