SCHEMBL527070

SCHEMBL527070

FC(F)C(F)Oc1ccncc1Br

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
CA14 Q9ULX7 1/20 0.33
CA1 P00915 2/20 0.32
AXL P30530 1/20 0.31
IKBKB O14920 1/20 0.31
CHUK O15111 1/20 0.31
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13724635 0.85 KDM4E (0.36) CA12CA2CA9CA14CA1
SCHEMBL28864446 0.78 AOC1 (0.37) CA12CA2CA9CA14CA1
SCHEMBL20481226 0.77 CA12 (0.37) CA12CA2CA9CA14CA1
SCHEMBL24200150 0.76 CA12 (0.36) CA12CA2CA9CA14CA1
SCHEMBL15777428 0.74 RORC (0.34) CA12CA2CA9CA14CA1
SCHEMBL15776169 0.74 CA12 (0.33) CA12CA2CA9CA14CA1
SCHEMBL28026353 0.74 RORC (0.34) CA12CA2CA9CA14CA1
SCHEMBL1400223 0.72 HTR1A (0.39)
SCHEMBL20190681 0.71 HTT (0.41) CHUK
SCHEMBL15475790 0.70 CA12 (0.33) CA12CA2CA9CA14CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598481-A1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS Bristol-Myers Squibb Company (US) 2013-06-05 EP disclosed
WO-2012015723-A1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-02 WO disclosed