SCHEMBL28026404

SCHEMBL28026404

COc1c(N)ccnc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
DYRK1A Q13627 1/20 0.42
NOS3 P29474 2/20 0.36
NOS2 P35228 2/20 0.36
NOS1 P29475 1/20 0.36
HASPIN Q8TF76 1/20 0.34
DYRK2 Q92630 1/20 0.34
ALOX5AP P20292 2/20 0.34
FEN1 P39748 2/20 0.34
LRRK2 Q5S007 1/20 0.34
AURKA O14965 2/20 0.33
AURKB Q96GD4 2/20 0.33
TTK P33981 1/20 0.33
INCENP Q9NQS7 1/20 0.33
GAK O14976 3/20 0.33
RIPK2 O43353 2/20 0.33
NLK Q9UBE8 2/20 0.33
EPHB6 O15197 1/20 0.33
ABL1 P00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4381004 0.79 SMN1; SMN2 (0.41) HTTHSD17B10DYRK1AGAKRIPK2
SCHEMBL23148039 0.78 DYRK1A (0.39) HTTHSD17B10DYRK1AHASPINDYRK2
SCHEMBL4380382 0.78 DYRK1A (0.39) HTTHSD17B10DYRK1ANOS3NOS2
SCHEMBL29813440 0.78 DYRK1A (0.39) HTTHSD17B10DYRK1AHASPINDYRK2
SCHEMBL8417801 0.76 AURKA (0.44) DYRK1ANOS3NOS2NOS1DYRK2
SCHEMBL29954197 0.75 DYRK1A (0.38) HTTHSD17B10DYRK1AHASPINDYRK2
SCHEMBL30050747 0.75 HTT (0.47) HTTHSD17B10DYRK1ANOS3NOS2
SCHEMBL29023076 0.75 HTT (0.47) HTTHSD17B10DYRK1ANOS3NOS2
SCHEMBL31602251 0.74 NOS2 (0.42) DYRK1ANOS3NOS2NOS1AURKA
SCHEMBL157196 0.74 HTT (0.50) HTTHSD17B10DYRK1ANOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104755465-A Heterocyclic compounds TAKEDA PHARMACEUTICAL 2015-07-01 CN disclosed