SCHEMBL28028156

SCHEMBL28028156

C=C(C#N)C(=O)OC(C(=O)NC1CC1)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)OC(=O)NCCOC(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 5/20 0.37
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
REN P00797 5/20 0.33
EDNRB P24530 2/20 0.33
EDNRA P25101 2/20 0.33
CTSD P07339 1/20 0.33
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
CTSK P43235 2/20 0.33
CTSS P25774 2/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
PSMB5 P28074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28028172 0.76 MEN1 (0.41) CAPN1MEN1TSHRKMT2AREN
SCHEMBL28028159 0.75 CAPN1 (0.46) CAPN1RENCTSKCTSSCTSL
SCHEMBL28821803 0.73 MEN1 (0.44) CAPN1MEN1TSHRKMT2ACTSD
SCHEMBL15299885 0.69 MEN1 (0.47) CAPN1MEN1TSHRKMT2AREN
SCHEMBL21457955 0.68 CAPN1 (0.61) CAPN1RENCTSKCTSL
SCHEMBL4391534 0.68 CAPN1 (0.61) CAPN1RENCTSKCTSL
SCHEMBL28028183 0.68 PSMB5 (0.37) RENCTSDCTSKPSMB5
SCHEMBL28027550 0.65 REN (0.40) RENCTSDPSMB5
SCHEMBL21458026 0.65 MEN1 (0.46) CAPN1MEN1TSHRKMT2AREN
SCHEMBL21555137 0.63 SMN1; SMN2 (0.45) CAPN1MEN1TSHRKMT2ACTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103282043-B Congenital agyria therapeutic agent OSAKA CITY UNIVERSITY (JP) 2015-09-30 CN disclosed