SCHEMBL28028536

SCHEMBL28028536

CC(CI)(N=C=O)c1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.38
RIPK1 Q13546 1/20 0.33
KIF11 P52732 1/20 0.33
HDAC6 Q9UBN7 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
CCR2 P41597 2/20 0.32
ACHE P22303 1/20 0.32
MIF P14174 1/20 0.31
CHRM3 P20309 1/20 0.31
PTPN1 P18031 1/20 0.31
MDM4 O15151 1/20 0.30
TP53 P04637 1/20 0.30
MDM2 Q00987 1/20 0.30
CETP P11597 1/20 0.30
TSHR P16473 1/20 0.30
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2572622 0.89 ESR1 (0.32) HDAC2ACHE
SCHEMBL28027917 0.80 CYP2C19 (0.36) HDAC6HDAC3HDAC1HDAC2TSHR
SCHEMBL25351936 0.78 GABRA1 (0.31)
SCHEMBL9585930 0.77 L3MBTL1 (0.41) TSHR
SCHEMBL4090896 0.74 GABRA1 (0.36) RIPK1HDAC2ACHE
SCHEMBL12501890 0.72 KCNN4 (0.32) KCNN4RIPK1HDAC6HDAC3HDAC1
SCHEMBL6555332 0.68
SCHEMBL2589886 0.68 PTGDR2 (0.31)
SCHEMBL18244101 0.67 KCNN4 (0.52) KCNN4RIPK1KIF11HDAC6HDAC3
SCHEMBL7929172 0.66 KCNN4 (0.50) KCNN4KIF11HDAC6HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958922-B 2,5,6,7-tetrahydrochysene-[Isosorbide-5-Nitrae] oxygen azepine *-3-base amine or 2,3,6,7-tetrahydrochysene-[Isosorbide-5-Nitrae] oxygen azepine *-5-ylamine compounds HOFFMAN-LA ROCHE LTD. (CH) 2015-09-30 CN disclosed