SCHEMBL28030656

SCHEMBL28030656

NC(=O)Cc1cccc(NC2CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.52
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
KCNH2 Q12809 1/20 0.46
CSNK2A1 P68400 1/20 0.44
F2RL1 P55085 1/20 0.42
SMYD3 Q9H7B4 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
AURKA O14965 2/20 0.40
EPHX2 P34913 1/20 0.40
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
CHEK1 O14757 1/20 0.39
MAP3K7 O43318 1/20 0.39
NUAK1 O60285 1/20 0.39
JAK2 O60674 1/20 0.39
BMX P51813 1/20 0.39
NEK2 P51955 1/20 0.39
MAP3K9 P80192 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17115656 0.84 SMN1; SMN2 (0.44) IRAK4OPRM1OPRD1OPRK1KCNH2
SCHEMBL15710125 0.82 MAPT (0.49) SMN1; SMN2KDM4ELMNA
SCHEMBL3184520 0.78 CSNK2A1 (0.49) CSNK2A1SMN1; SMN2AURKAEPHX2CHEK1
SCHEMBL15387062 0.77 CSNK2A1 (0.48) CSNK2A1SMN1; SMN2AURKAEPHX2CHEK1
SCHEMBL11627789 0.77 CSNK2A1 (0.54) CSNK2A1SMN1; SMN2AURKALMNA
SCHEMBL14148255 0.77 CSNK2A1 (0.48) CSNK2A1SMN1; SMN2AURKACHEK1MAP3K7
SCHEMBL30401772 0.76 CRBN (0.74) DDB1CRBN
SCHEMBL10339219 0.75 CA2 (0.54) CSNK2A1KDM4ELMNA
SCHEMBL13920446 0.75 DDB1 (0.49) IRAK4OPRM1OPRD1OPRK1KCNH2
SCHEMBL5037396 0.74 ALDH1A1 (0.57) CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104936954-A compounds and methods of use thereof AGIOS PHARMACEUTICALS INC 2015-09-23 CN disclosed