SCHEMBL28031300

SCHEMBL28031300

Nc1ccc2nc(-c3cccnc3)ncc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
HTT P42858 3/20 0.52
AXL P30530 2/20 0.50
MEN1 O00255 1/20 0.50
PSIP1 O75475 1/20 0.50
MKNK1 Q9BUB5 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
ABCG2 Q9UNQ0 2/20 0.48
LMNA P02545 3/20 0.48
POLB P06746 1/20 0.48
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
TP53 P04637 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HSD17B10 Q99714 2/20 0.47
HSP90AA1 P07900 2/20 0.47
HSP90AB1 P08238 2/20 0.47
TSHR P16473 2/20 0.47
CASP1 P29466 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28031380 0.88 AXL (0.50) MAPTHTTAXLMEN1PSIP1
SCHEMBL3191937 0.84 TLR9 (0.57) MAPTHTTMEN1LMNAALDH1A1
SCHEMBL27887749 0.82 CYP2A6 (0.47) MAPTHTTMEN1LMNAPOLB
SCHEMBL27483583 0.79 CYP2A6 (0.56) MAPTHTTMEN1LMNAPOLB
SCHEMBL14906702 0.77 CYP2A6 (0.67) MAPTHTTAXLMEN1PSIP1
SCHEMBL14474112 0.75 GBA1 (0.41) MAPTHTTMEN1LMNAALDH1A1
SCHEMBL7601945 0.75 EGFR (0.45) MAPTHTTMEN1LMNAPOLB
SCHEMBL15617051 0.75 CYP2A6 (0.69) MAPTHTTAXLMEN1PSIP1
SCHEMBL24335889 0.74 PIK3CA (0.55) MAPTHTTAXLMEN1PSIP1
SCHEMBL2239546 0.73 NPC1 (0.50) MAPTHTTMEN1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105218516-A Therapeutic compounds and related methods of use OTSUKA PHARMA CO LTD 2016-01-06 CN disclosed
CN-102883723-B Therapeutic compounds and related methods of use OTSUKA PHARMACEUTICAL CO.,LTD. (JP) 2015-09-16 CN disclosed