SCHEMBL2803161

SCHEMBL2803161

CC(C)Nc1nc(-c2ccco2)nc2ccc(I)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.47
ACP1 P24666 1/20 0.45
KDM1A O60341 1/20 0.43
GBA1 P04062 2/20 0.42
GGPS1 O95749 1/20 0.39
ADORA3 P0DMS8 6/20 0.39
ADORA2A P29274 4/20 0.39
ADORA1 P30542 3/20 0.39
ADORA2B P29275 1/20 0.38
CCNE2 O96020 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
APP P05067 1/20 0.37
CSNK1A1 P48729 1/20 0.37
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37
HTR3A P46098 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
LATS1 O95835 1/20 0.36
LATS2 Q9NRM7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13088248 0.82 PDE5A (0.47) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL3811994 0.81 PDE5A (0.46) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL2804534 0.80 ACP1 (0.45) PDE5AACP1KDM1AGBA1ADORA3
SCHEMBL30772425 0.78 PDE5A (0.41) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL2803755 0.78 PDE5A (0.41) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL2803607 0.77 PDE5A (0.40) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL2803611 0.77 PDE5A (0.40) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL2802463 0.77 PDE5A (0.44) PDE5AKDM1AGBA1ADORA3ADORA2A
SCHEMBL2806792 0.75 PDE5A (0.38) PDE5AACP1KDM1AGBA1GGPS1
SCHEMBL2806796 0.75 PDE5A (0.38) PDE5AACP1KDM1AGBA1GGPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2241565-A1 Aurora kinase inhibitors compounds Universität Leipzig (DE) 2010-10-20 EP disclosed
EP-2241565-A1 Aurora kinase inhibitors compounds Universität Leipzig (DE) 2010-10-20 EP disclosed
WO-2010081881-A1 AURORA KINASE INHIBITORS COMPOUNDS. UNIVERSITÄT LEIPZIG (DE) 2010-07-22 WO disclosed
WO-2010081881-A1 AURORA KINASE INHIBITORS COMPOUNDS. UNIVERSITÄT LEIPZIG (DE) 2010-07-22 WO disclosed