SCHEMBL28032226

SCHEMBL28032226

COC(=O)c1c(-c2ccccc2)cn(-c2ccc(OC)cc2)c1C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.44
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.43
TDP1 Q9NUW8 1/20 0.43
PTPN11 Q06124 3/20 0.43
GABRA1 P14867 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43
GABRA2 P47869 1/20 0.43
MAPT P10636 4/20 0.42
PKM P14618 1/20 0.42
LMNA P02545 2/20 0.42
TP53 P04637 2/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28031629 0.93 KDM4E (0.47) GFERKDM4EALDH1A1TDP1PTPN11
SCHEMBL28194102 0.90 MEN1 (0.43) KDM4EALDH1A1GABRA1GABRG2GABRB3
SCHEMBL28031631 0.90 PTPN11 (0.47) GFERKDM4EALDH1A1TDP1PTPN11
SCHEMBL28031707 0.85 ALDH1A1 (0.46) GFERKDM4EALDH1A1TDP1PTPN11
SCHEMBL28031643 0.83 MEN1 (0.44) KDM4EALDH1A1TDP1GABRA1GABRG2
SCHEMBL28078513 0.81 MEN1 (0.49) KDM4EALDH1A1TDP1GABRA1GABRG2
SCHEMBL28078523 0.81 PDE5A (0.39) GFERKDM4EALDH1A1PTPN11MAPT
SCHEMBL28931713 0.80 MEN1 (0.58) GFERKDM4EALDH1A1TDP1GABRA1
SCHEMBL28032234 0.80 MEN1 (0.45) KDM4EALDH1A1PTPN11GABRA1GABRG2
SCHEMBL28031775 0.79 TP53 (0.45) GFERKDM4EALDH1A1PTPN11GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017126-B Perfluoroalkyl azole derivatives and its synthetic method 上海麦克林生化科技有限公司 2018-01-19 CN disclosed
CN-105017126-A Perfluoroalkyl pyrrole derivative and synthesis method thereof UNIV SHANGHAI 2015-11-04 CN disclosed