SCHEMBL28032448

SCHEMBL28032448

[c]1c[nH]c2cc(CCN3CCOCC3)ccc12

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.54
L3MBTL3 Q96JM7 1/20 0.40
POLB P06746 1/20 0.39
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
HRH3 Q9Y5N1 1/20 0.36
SLC6A4 P31645 1/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016009 0.85 TNKS2 (0.47) POLBCYP1A2CYP2D6PARP1
SCHEMBL6016018 0.78 KDM4E (0.55) SIGMAR1KCNH2CYP1A2HRH3
SCHEMBL27601537 0.76 SLC6A2 (0.38) SIGMAR1CYP2D6SLC6A4
SCHEMBL6015810 0.73 ALDH1A1 (0.60) POLBCYP2D6
SCHEMBL6016002 0.73 ATM (0.58) CYP1A2HRH3
SCHEMBL6015767 0.73 POLB (0.60) POLBKCNH2CYP1A2CYP2D6PARP1
SCHEMBL6015785 0.70 ALDH1A1 (0.55) SIGMAR1KCNH2CYP1A2HRH3PARP1
SCHEMBL15987537 0.70 SIGMAR1 (0.56) SIGMAR1L3MBTL3POLBKCNJ1KCNH2
SCHEMBL3176117 0.69 SIGMAR1 (0.63) SIGMAR1L3MBTL3POLBCYP1A2CYP2D6
SCHEMBL3186832 0.69 SIGMAR1 (0.55) SIGMAR1L3MBTL3POLBCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104936596-A Neuroprotective CB2 receptor agonists CLEVELAND CLINIC FOUNDATION 2015-09-23 CN disclosed