SCHEMBL28032867

SCHEMBL28032867

CN1CCN(CCCOc2ccc3cncnc3c2)CC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.62
DRD3 P35462 3/20 0.62
EGFR P00533 1/20 0.52
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
HRH1 P35367 1/20 0.48
USP2 O75604 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
HRH4 Q9H3N8 3/20 0.47
SIGMAR1 Q99720 1/20 0.46
XDH P47989 2/20 0.45
CXCR1 P25024 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18128966 0.94 EGFR (0.54) HRH3DRD3EGFRUSP2ALDH1A1
SCHEMBL28032396 0.90 HRH3 (0.62) HRH3DRD3EGFRNPC1RAB9A
SCHEMBL7837580 0.90 HRH3 (0.53) HRH3EGFR
SCHEMBL5680969 0.89 HRH3 (0.55) HRH3
SCHEMBL3067381 0.86 HRH3 (0.54) HRH3EGFRHRH1USP2ALDH1A1
SCHEMBL30979868 0.86 HRH3 (0.54) HRH3EGFRHRH1USP2ALDH1A1
SCHEMBL30209183 0.86 HRH3 (0.49) HRH3DRD3EGFRHRH1ALDH1A1
SCHEMBL6689692 0.86 HRH3 (0.45) HRH3DRD3EGFRHRH1
SCHEMBL5679317 0.86 HRH3 (0.45) HRH3DRD3EGFRHRH1SIGMAR1
SCHEMBL10807692 0.83 HRH3 (0.70) HRH3DRD3NPC1RAB9AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101090899-B 2,5 and 2,6 disubstituted benzazole analogs useful as protein kinase inhibitors 4SC Corp. (DE) 2015-09-09 CN disclosed