SCHEMBL28033009

SCHEMBL28033009

CCn1c(CCCCC(=O)O)nc2c1c(=O)n(C)c(=O)n2C

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.59
ALOX15 P16050 1/20 0.59
ALDH1A1 P00352 3/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 2/20 0.54
TSHR P16473 2/20 0.53
HTT P42858 1/20 0.50
PDE4B Q07343 1/20 0.48
NCOA1 Q15788 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
RECQL P46063 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 1/20 0.47
HSD17B10 Q99714 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28064034 0.88 CYP1A2 (0.57) ALDH1A1CYP1A2CYP2C19KMT2ARXFP1
SCHEMBL28033007 0.88 ALDH1A1 (0.50) MAPK1ALOX15ALDH1A1CYP1A2CYP2C19
SCHEMBL28033011 0.86 CYP2C19 (0.47) MAPK1ALOX15ALDH1A1CYP1A2CYP2C19
SCHEMBL28033489 0.85 ALOX15 (0.63) MAPK1ALOX15ALDH1A1TSHRHTT
SCHEMBL19969448 0.76 RXFP1 (0.59) CYP2C19KMT2ARXFP1
Dimethylamine SCHEMBL11384972 0.75 TSHR (0.61) MAPK1ALOX15ALDH1A1CYP1A2CYP2C19
SCHEMBL19969451 0.74 RXFP1 (0.57) CYP2C19KMT2ARXFP1
Dimethylamine SCHEMBL11379643 0.74 TSHR (0.60) MAPK1ALOX15ALDH1A1CYP1A2CYP2C19
SCHEMBL683896 0.72 TSHR (0.56) MAPK1ALOX15ALDH1A1CYP1A2CYP2C19
Diethylamine SCHEMBL11380621 0.72 TSHR (0.57) MAPK1ALOX15ALDH1A1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104892610-A Preparation method of 8-ester based caffeine derivative UNIV FUJIAN 2015-09-09 CN disclosed