SCHEMBL28064034

SCHEMBL28064034

Cn1c(=O)c2c(nc(CCCCC(=O)O)n2C)n(C)c1=O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.57
CYP2C19 P33261 2/20 0.57
ALDH1A1 P00352 1/20 0.57
RXFP1 Q9HBX9 2/20 0.52
MAOB P27338 3/20 0.49
MAOA P21397 2/20 0.49
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19969448 0.88 RXFP1 (0.59) CYP2C19RXFP1MAOBMAOAKMT2A
SCHEMBL28033009 0.88 MAPK1 (0.59) CYP1A2CYP2C19ALDH1A1RXFP1KMT2A
SCHEMBL28033011 0.87 CYP2C19 (0.47) CYP1A2CYP2C19ALDH1A1
SCHEMBL19969451 0.87 RXFP1 (0.57) CYP2C19RXFP1MAOBMAOAKMT2A
SCHEMBL28033007 0.84 ALDH1A1 (0.50) CYP1A2CYP2C19ALDH1A1KMT2A
SCHEMBL25155042 0.83 RXFP1 (0.51) CYP2C19ALDH1A1RXFP1MAOBMAOA
SCHEMBL26439802 0.83 RXFP1 (0.51) CYP2C19ALDH1A1RXFP1MAOBMAOA
SCHEMBL19969447 0.82 RXFP1 (0.62) CYP2C19RXFP1MAOBMAOAKMT2A
SCHEMBL28033489 0.81 ALOX15 (0.63) ALDH1A1
SCHEMBL15071609 0.81 CYP1A2 (0.56) CYP1A2CYP2C19RXFP1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104892610-B A kind of preparation method of 8-ester group caffeine derivative 福建师范大学 2016-08-24 CN disclosed