SCHEMBL28036047

SCHEMBL28036047

CCOC(=O)CC(C(C)=O)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.46
MGAM O43451 1/20 0.46
SI P14410 1/20 0.46
MGAM2 Q2M2H8 1/20 0.46
ALDH1A1 P00352 7/20 0.43
TRPA1 O75762 1/20 0.43
HSD17B10 Q99714 2/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 2/20 0.40
ALOX15 P16050 3/20 0.40
CYP3A4 P08684 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
CHRM1 P11229 1/20 0.39
ADORA1 P30542 1/20 0.39
CYP1A2 P05177 1/20 0.38
SOAT1 P35610 1/20 0.36
CYP2D6 P10635 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
HCAR2 Q8TDS4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1194353 0.91 GAA (0.50) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL8917503 0.89 ALDH1A1 (0.54) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL460011 0.87 MGAM (0.46) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL12877143 0.83 GAA (0.48) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL23071556 0.83 HCAR2 (0.38) ALDH1A1LMNATSHRTDP1CHRM1
SCHEMBL17053359 0.83 MGAM (0.43) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL14485615 0.82 MGAM (0.41) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL27703510 0.80 MGAM (0.45) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL3326034 0.80 MGAM (0.40) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL430204 0.79 MGAM (0.52) GAAMGAMSIMGAM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189511-A Inhibitors of human immunodeficiency virus replication BRISTOL MYERS SQUIBB CO 2015-12-23 CN disclosed
CN-105189510-A Inhibitors of human immunodeficiency virus replication BRISTOL MYERS SQUIBB CO 2015-12-23 CN disclosed
CN-105008369-A INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL MYERS SQUIBB CO 2015-10-28 CN disclosed