SCHEMBL28036649

SCHEMBL28036649

COC(=O)CC[C@@H](COS(=O)(=O)c1ccc(CN)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 12/20 0.40
MAPT P10636 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
PKM P14618 2/20 0.38
HPGD P15428 2/20 0.38
TSHR P16473 2/20 0.38
HTT P42858 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TP53 P04637 1/20 0.38
AGTR1 P30556 1/20 0.38
RAB9A P51151 1/20 0.38
CA1 P00915 7/20 0.38
CA9 Q16790 2/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
PTPRB P23467 2/20 0.36
ATM Q13315 2/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL384396 0.89 ALDH1A1 (0.42) CA2MAPTALDH1A1LMNAPKM
SCHEMBL12944323 0.83 ALDH1A1 (0.43) CA2MAPTALDH1A1LMNAPKM
SCHEMBL3089832 0.79 ALDH1A1 (0.45) CA2ALDH1A1TSHRCA1CA9
SCHEMBL28968914 0.79 ALDH1A1 (0.45) CA2ALDH1A1TSHRCA1CA9
SCHEMBL30096737 0.78 ALDH1A1 (0.41) CA2MAPTALDH1A1LMNAPKM
SCHEMBL30096762 0.78 ALDH1A1 (0.41) CA2MAPTALDH1A1LMNAPKM
SCHEMBL22006099 0.78 CA2 (0.40) CA2MAPTALDH1A1LMNAPKM
SCHEMBL29255200 0.74 ALDH1A1 (0.42) CA2ALDH1A1LMNAPKMTSHR
SCHEMBL8193095 0.74 ALDH1A1 (0.43) CA2ALDH1A1LMNAPKMHPGD
SCHEMBL25022221 0.73 CA2 (0.41) CA2TSHRCA1CA7ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103351389-B Aminopurine, its composition that halogenated aryl replaces, and use it for the method for the treatment of SIGNAL PHARM LLC (US) 2015-10-28 CN disclosed