SCHEMBL28036688

SCHEMBL28036688

COc1c(O)cccc1-c1ccc(N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
USP7 Q93009 1/20 0.40
APP P05067 1/20 0.40
TP53 P04637 2/20 0.39
TSHR P16473 1/20 0.39
CDK4 P11802 1/20 0.39
CCNA2 P20248 1/20 0.39
CCND1 P24385 1/20 0.39
CDK2 P24941 1/20 0.39
CCND3 P30281 1/20 0.39
PDE4B Q07343 3/20 0.39
PDE4A P27815 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
TUBB4A P04350 3/20 0.38
TUBB P07437 3/20 0.38
TUBA3C P0DPH7 3/20 0.38
TUBA1B P68363 3/20 0.38
TUBA4A P68366 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL526920 0.83 ALDH1A1 (0.56) CA1CA2TP53TSHRCDK4
SCHEMBL29431716 0.83 ALDH1A1 (0.56) CA1CA2TP53TSHRCDK4
SCHEMBL28314094 0.82 SLC6A4 (0.46) CA1CA2TP53TSHRCDK4
SCHEMBL3786304 0.81 FYN (0.42) APPTP53CDK4CCND1CDK2
SCHEMBL21815270 0.80 CA1 (0.55) CA1CA2TP53TSHRCDK2
SCHEMBL28222892 0.80 CYP19A1 (0.53) TP53TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL22777983 0.79 PRKAB2 (0.52) CA1CA2APPTP53TSHR
SCHEMBL6132279 0.79 MME (0.43) APPTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL29869241 0.79 IKBKB (0.43) CA1CA2TP53CDK4CCNA2
SCHEMBL6011377 0.78 CA1 (0.40) CA1CA2TP53TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017056-B Phenylpropen ketone derivatives and its preparation method and pharmaceutical composition and purposes 中国医学科学院药物研究所 2019-02-01 CN disclosed
CN-105017056-A Phenyl acrylketone derivative and preparation method, drug composition and application thereof INST MATERIA MEDICA CAMS 2015-11-04 CN disclosed