SCHEMBL28037155

SCHEMBL28037155

C#Cc1ccc(N2CCC(C)CC2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 3/20 0.45
MAPK1 P28482 2/20 0.45
MAPT P10636 2/20 0.45
AR P10275 1/20 0.43
HTT P42858 1/20 0.42
CYP2C9 P11712 1/20 0.41
HPGD P15428 3/20 0.40
HSD17B10 Q99714 2/20 0.39
DPP4 P27487 1/20 0.39
GAA P10253 4/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.38
NR4A1 P22736 1/20 0.38
HSD11B1 P28845 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037584 0.84 NOTUM (0.47) ARPDE3BPDE3ANOTUM
SCHEMBL15122274 0.81 NOTUM (0.51) ALDH1A1KDM4EMAPTGAAPOLB
SCHEMBL28037158 0.81 NCF1 (0.45) ALDH1A1KDM4EMAPTCYP2C9NOTUM
SCHEMBL29722987 0.78 ALDH1A1 (0.65) ALDH1A1KDM4EMAPK1MAPTAR
SCHEMBL853170 0.78 ALDH1A1 (0.65) ALDH1A1KDM4EMAPK1MAPTAR
SCHEMBL13175782 0.76 AR (0.51) ALDH1A1ARHTTDPP4GAA
SCHEMBL1963730 0.75 DPP4 (0.56) ALDH1A1KDM4EMAPTARDPP4
SCHEMBL23648678 0.73 PDE3B (0.50) ALDH1A1MAPTCYP2C9DPP4MEN1
SCHEMBL20578110 0.73 GAA (0.67) ALDH1A1KDM4EMAPTHTTCYP2C9
SCHEMBL8261930 0.72 CTPS1 (0.62) ALDH1A1KDM4EMAPK1MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105061326-A Pyridazinone derivatives as well as preparation method and application thereof SICHUAN BAILI PHARMACEUTICAL CO LTD 2015-11-18 CN disclosed