SCHEMBL28037273

SCHEMBL28037273

Cn1ccc(-c2ccc(C#N)cc2)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.58
KMT2A Q03164 1/20 0.57
CYP19A1 P11511 1/20 0.51
SCN4A P35499 1/20 0.49
GAA P10253 1/20 0.46
CYP11B2 P19099 3/20 0.45
CHEK1 O14757 2/20 0.43
F2RL3 Q96RI0 1/20 0.42
EP300 Q09472 1/20 0.42
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2C P18825 1/20 0.41
HTR1D P28221 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR7 P34969 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KIF11 P52732 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8807623 0.79 GRM5 (0.58) KMT2A
SCHEMBL6852707 0.78 KEAP1 (0.55) KEAP1KMT2ACYP19A1SCN4ACHEK1
SCHEMBL26199262 0.76 SCN4A (0.52) KEAP1KMT2ACYP19A1SCN4ACYP11B2
SCHEMBL12319225 0.75 KEAP1 (0.67) KEAP1KMT2ACYP19A1SCN4AGAA
SCHEMBL15885116 0.75 CHEK1 (0.56) KEAP1KMT2ACYP19A1SCN4ACHEK1
SCHEMBL28734542 0.75 ALDH1A1 (0.48) KMT2AGAACYP11B2CHEK1NPC1
SCHEMBL17090942 0.74 CYP19A1 (0.50) CYP19A1GAACYP11B2CHEK1F2RL3
SCHEMBL28037403 0.74 GAA (0.41) GAACHEK1F2RL3NPC1RAB9A
SCHEMBL6847795 0.74 KEAP1 (0.50) KEAP1KMT2ACYP19A1SCN4ACHEK1
SCHEMBL15885670 0.74 KEAP1 (0.64) KEAP1KMT2ACYP19A1SCN4ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164124-B Compounds and compositions for treating parasitic diseases 诺华股份有限公司 2017-03-15 CN disclosed
CN-105164124-A Compounds and compositions for treating parasitic diseases NOVARTIS AG 2015-12-16 CN disclosed