SCHEMBL28038757

SCHEMBL28038757

COc1c(Cl)cccc1C1CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
TAS1R3 Q7RTX0 2/20 0.40
TAS1R1 Q7RTX1 2/20 0.40
TAS1R2 Q8TE23 2/20 0.40
HTR2C P28335 2/20 0.40
SLC6A3 Q01959 4/20 0.39
HTR1A P08908 3/20 0.39
SLC6A2 P23975 3/20 0.39
SLC6A4 P31645 3/20 0.39
ADRA1A P35348 1/20 0.38
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
GRIA1 P42261 1/20 0.37
CACNG8 Q8WXS5 1/20 0.37
ATM Q13315 1/20 0.37
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
OPRL1 P41146 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19703133 0.88 HTR2C (0.57) HTR2CSLC6A3HTR1ASLC6A2SLC6A4
SCHEMBL22062953 0.87 MEN1 (0.46) MEN1KMT2ATAS1R3TAS1R1TAS1R2
SCHEMBL27845122 0.81 CA1 (0.46) MEN1KMT2ATAS1R3TAS1R1TAS1R2
SCHEMBL8109922 0.78 HTR2C (0.41) MEN1KMT2AHTR2CSLC6A3HTR1A
SCHEMBL29639264 0.78 HTR2C (0.53) MEN1KMT2AHTR2CSLC6A3HTR1A
SCHEMBL16951549 0.78 HTR2C (0.46) HTR2CSLC6A3HTR1ASLC6A2SLC6A4
SCHEMBL7779150 0.78 MEN1 (0.35) MEN1KMT2ATAS1R3TAS1R1TAS1R2
SCHEMBL4439192 0.78 NOTUM (0.39) KMT2ATAS1R3TAS1R1TAS1R2SLC6A3
SCHEMBL2046629 0.77 HTR1A (0.50) HTR2CSLC6A3HTR1ASLC6A2SLC6A4
SCHEMBL28092534 0.77 HTR2C (0.43) HTR2CSLC6A3HTR1ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103097364-B Spiro-piperidine derivatives as S1P modulators ABBOTT HEALTHCARE PRODUCTS B.V. (NL) 2015-11-25 CN disclosed