SCHEMBL28039291

SCHEMBL28039291

Cc1cc(C(=O)O)cc(C(=O)O)c1.O=C(O)c1cn(-c2ccccc2)nn1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 4/20 0.49
L3MBTL1 Q9Y468 2/20 0.46
POLB P06746 1/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA4 P22748 2/20 0.45
CA9 Q16790 2/20 0.45
HPGDS O60760 1/20 0.44
ALKBH2 Q6NS38 1/20 0.44
NOTUM Q6P988 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
MIF P14174 1/20 0.44
TPMT P51580 1/20 0.43
P2RX7 Q99572 1/20 0.42
KMT2A Q03164 1/20 0.42
RIPK1 Q13546 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL69876 0.85 ESRRA (0.62) ESRRAL3MBTL1CA1CA2CA4
SCHEMBL28801446 0.83 ESRRA (0.60) ESRRAL3MBTL1CA1CA2CA4
SCHEMBL69165 0.81 ESRRA (0.64) ESRRACA1CA2CA9MAOA
SCHEMBL3477570 0.81 CA1 (0.57) ESRRAL3MBTL1POLBCA1CA2
SCHEMBL27498827 0.79 CYP2C9 (0.47) L3MBTL1HPGDSALKBH2TPMTKMT2A
SCHEMBL27575419 0.77 ALKBH2 (0.77) HPGDSALKBH2KMT2A
SCHEMBL31734379 0.77 HPGDS (0.57) ESRRAL3MBTL1CA1CA2CA4
SCHEMBL1749529 0.76 OGT (0.53) ESRRACA1CA2CA4CA9
SCHEMBL28167460 0.76 NOTUM (0.53) L3MBTL1POLBHPGDSALKBH2NOTUM
SCHEMBL23889183 0.76 ESRRA (0.59) ESRRAL3MBTL1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073741-A Phthalazinones and isoquinolinones as rock inhibitors BRISTOL MYERS SQUIBB CO 2015-11-18 CN disclosed