SCHEMBL28801446

SCHEMBL28801446

O=C(O)c1cn(-c2ccccc2)nn1.[LiH]

nearest known ligand 0.77

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 5/20 0.60
P2RX7 Q99572 1/20 0.53
NOTUM Q6P988 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA4 P22748 2/20 0.51
CA9 Q16790 2/20 0.51
RIPK1 Q13546 1/20 0.50
MAOA P21397 1/20 0.47
HPGDS O60760 1/20 0.47
ALKBH2 Q6NS38 1/20 0.47
SPR P35270 1/20 0.46
NPC1 O15118 1/20 0.46
MIF P14174 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL69876 0.98 ESRRA (0.62) ESRRAP2RX7NOTUML3MBTL1CA1
SCHEMBL31734379 0.89 HPGDS (0.57) ESRRAP2RX7NOTUML3MBTL1CA1
SCHEMBL1749529 0.88 OGT (0.53) ESRRACA1CA2CA4CA9
SCHEMBL27768462 0.87 ESRRA (0.71) ESRRAP2RX7NOTUML3MBTL1CA1
SCHEMBL23889183 0.84 ESRRA (0.59) ESRRAP2RX7NOTUML3MBTL1CA1
SCHEMBL19691104 0.84 ESRRA (0.63) ESRRAP2RX7NOTUML3MBTL1CA1
SCHEMBL27877288 0.84 ESRRA (0.57) ESRRACA1CA2CA4CA9
SCHEMBL23153549 0.84 ESRRA (0.59) ESRRAP2RX7NOTUML3MBTL1CA1
SCHEMBL4708257 0.84 MAOA (0.49) ESRRANOTUML3MBTL1CA1CA2
SCHEMBL28039291 0.83 ESRRA (0.49) ESRRAP2RX7NOTUML3MBTL1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102985439-B9 IAP BIR domain binding compounds 制药科学股份有限公司 2016-08-03 CN disclosed
CN-102985439-B IAP BIR domain binding compounds 制药科学股份有限公司 2016-06-15 CN disclosed
CN-102985439-A IAP BIR domain binding compounds AEGERA THERAPEUTICS INC 2013-03-20 CN disclosed