SCHEMBL28039299

SCHEMBL28039299

COc1cc(OC)cc(-c2nccn2C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 6/20 0.44
CYP1A1 P04798 5/20 0.44
CYP1A2 P05177 3/20 0.42
CYP2E1 P05181 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C8 P10632 3/20 0.42
CYP2D6 P10635 3/20 0.42
CYP2A6 P11509 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP4B1 P13584 3/20 0.42
CYP2B6 P20813 3/20 0.42
CYP3A5 P20815 3/20 0.42
CYP2A7 P20853 3/20 0.42
CYP3A7 P24462 3/20 0.42
CYP2F1 P24903 3/20 0.42
CYP2C18 P33260 3/20 0.42
CYP2C19 P33261 3/20 0.42
CYP2J2 P51589 3/20 0.42
CYP4F2 P78329 3/20 0.42
CYP4F8 P98187 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362756 0.83 DYRK1A (0.56) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL13052883 0.82 LPO (0.46) KDM4ENPC1RAB9A
SCHEMBL14675684 0.81 CLK4 (0.48) CYP3A4CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL24575918 0.80 CCR1 (0.41) CYP1B1CYP1A1CYP1A2CYP2E1CYP3A4
SCHEMBL16131408 0.76 LPO (0.46) HPGDKDM4ENPC1RAB9A
SCHEMBL4259944 0.74 CCR1 (0.61) POLBDYRK1ANPC1RAB9A
SCHEMBL23571873 0.74 F2 (0.49) ALDH1A1POLBDYRK1ACLK4
SCHEMBL28050431 0.74 LRRK2 (0.51) ALDH1A1HPGDKDM4EMAPTCCNB2
SCHEMBL12320472 0.73 LPO (0.39) KDM4ENPC1RAB9A
SCHEMBL31398200 0.73 LPO (0.39) ALDH1A1KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164125-B 2-phenyl or 2-heteroaryl imidazo [1,2-a ] pyridine derivatives 豪夫迈·罗氏有限公司 2017-10-13 CN claimed
CN-105229009-B 2-phenylimidazo [1,2-A ] pyrimidines as imaging agents 豪夫迈·罗氏有限公司 2017-09-29 CN claimed
CN-105229009-A 2-phenylimidazo [1,2-A ] pyrimidines as imaging agents HOFFMANN LA ROCHE 2016-01-06 CN claimed
CN-105164125-A 2-phenyl or 2-heteroaryl imidazo [1, 2-a ] pyridine derivatives HOFFMANN LA ROCHE 2015-12-16 CN claimed
CN-105164125-B 2-phenyl or 2-heteroaryl imidazo [1,2-a ] pyridine derivatives 豪夫迈·罗氏有限公司 2017-10-13 CN disclosed
CN-105229009-B 2-phenylimidazo [1,2-A ] pyrimidines as imaging agents 豪夫迈·罗氏有限公司 2017-09-29 CN disclosed
CN-105229009-A 2-phenylimidazo [1,2-A ] pyrimidines as imaging agents HOFFMANN LA ROCHE 2016-01-06 CN disclosed
CN-105164125-A 2-phenyl or 2-heteroaryl imidazo [1, 2-a ] pyridine derivatives HOFFMANN LA ROCHE 2015-12-16 CN disclosed