SCHEMBL28039585

SCHEMBL28039585

CC(=O)Oc1n[nH]c2cc(F)ccc12

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 13/20 0.51
MAPK1 P28482 3/20 0.49
MAPK6 Q16659 2/20 0.49
MAP2K7 O14733 2/20 0.42
MAPKAPK2 P49137 1/20 0.41
MAPKAPK3 Q16644 1/20 0.41
AMY1A P0DUB6 1/20 0.40
ITK Q08881 3/20 0.40
GSK3B P49841 1/20 0.40
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27677673 0.88 MAP2K4 (0.42) MAP2K4MAPK1MAPK6AMY1AITK
SCHEMBL28776088 0.82 DYRK1A (0.57) GSK3B
SCHEMBL6612570 0.82 MAP2K4 (0.51) MAP2K4MAPK1AMY1AGSK3B
SCHEMBL1573919 0.78 HRH4 (0.47) MAP2K4MAPK1MAPK6HTR2A
SCHEMBL1574410 0.78 MAP2K4 (0.46) MAP2K4MAPK1MAPK6
SCHEMBL5820415 0.78 KDM4E (0.53) MAP2K4GSK3B
SCHEMBL1573862 0.77 ALDH1A1 (0.44) MAP2K4MAPK1MAPK6HTR2A
SCHEMBL1573971 0.77 MAP2K4 (0.42) MAP2K4MAPK1MAPK6GSK3BHTR2A
SCHEMBL1573835 0.76 GAA (0.45) MAP2K4MAPK1MAPK6HTR2A
SCHEMBL1573879 0.75 MAP2K4 (0.41) MAP2K4MAPK1MAPK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073741-A Phthalazinones and isoquinolinones as rock inhibitors BRISTOL MYERS SQUIBB CO 2015-11-18 CN disclosed