SCHEMBL28040340

SCHEMBL28040340

Cc1nc(Sc2ccc(N)cc2)sc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 4/20 0.43
RAB9A P51151 4/20 0.43
GAA P10253 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TSHR P16473 2/20 0.42
HPGD P15428 2/20 0.42
NPC1 O15118 3/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.37
HSP90AA1 P07900 1/20 0.36
PKM P14618 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM1A O60341 1/20 0.36
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
TARBP2 Q15633 1/20 0.35
GABRP O00591 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4919985 0.86 SMN1; SMN2 (0.55) SMN1; SMN2KDM4ERAB9AGAAALDH1A1
SCHEMBL10667681 0.78 CYP3A4 (0.45) SMN1; SMN2RAB9ATSHRNPC1KMT2A
SCHEMBL14018508 0.74 RAB9A (0.77) SMN1; SMN2KDM4ERAB9AGAAALDH1A1
SCHEMBL10360761 0.73 ALDH1A1 (0.57) SMN1; SMN2KDM4ERAB9AGAAALDH1A1
SCHEMBL28040345 0.72 HTT (0.46) SMN1; SMN2KDM4EALDH1A1TSHRHPGD
SCHEMBL4493748 0.70 ALDH1A1 (0.58) SMN1; SMN2KDM4ERAB9AALDH1A1HPGD
SCHEMBL11392854 0.68 ALDH1A1 (0.50) SMN1; SMN2KDM4ERAB9AGAAALDH1A1
SCHEMBL179966 0.68 ALDH1A1 (0.63) SMN1; SMN2KDM4ERAB9AGAAALDH1A1
SCHEMBL9748472 0.67 ALDH1A1 (0.54) SMN1; SMN2KDM4ERAB9AGAAALDH1A1
SCHEMBL11588944 0.67 MAPT (0.43) KDM4ERAB9AGAAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085482-B Substituted diethylenediamine compound and its application method and purposes 广东东阳光药业有限公司 2018-08-10 CN disclosed
CN-105085482-A Substituted piperazine compound, and usage method and application thereof GUANGDONG HEC PHARMACEUTICAL 2015-11-25 CN disclosed