SCHEMBL28041177

SCHEMBL28041177

c1cc(OCC2CC2)ccn1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 4/20 0.50
PARP10 Q53GL7 4/20 0.50
PARP2 Q9UGN5 2/20 0.50
TDP1 Q9NUW8 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
KDM1A O60341 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17321283 0.92 PARP15 (0.53) PARP15PARP10PARP2TDP1
SCHEMBL31680768 0.87 PARP15 (0.44) PARP15PARP10PARP2TDP1SIGMAR1
SCHEMBL15204083 0.87 TDP1 (0.63) TDP1KDM1A
SCHEMBL12525730 0.87 SLC2A1 (0.46) PARP15PARP10PARP2TDP1KDM1A
Hydrochloric Acid SCHEMBL2566398 0.85 TDP1 (0.66) TDP1KDM1A
SCHEMBL29024848 0.84 PARP15 (0.64) PARP15PARP10PARP2TDP1SIGMAR1
SCHEMBL28289262 0.79 NFE2L2 (0.51)
SCHEMBL1990800 0.77 TDP1 (0.57) PARP15PARP10PARP2TDP1
Water SCHEMBL27540910 0.77 PARP15 (0.53) PARP15PARP10PARP2TDP1SIGMAR1
SCHEMBL10280025 0.76 CHRNB2 (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107501274-B It can be used as the compound of ATR kinase inhibitor Votex Pharmaceutical Co., Ltd. (US) 2019-11-22 CN disclosed
CN-107501275-B It can be used as the compound of ATR kinase inhibitor Votex Pharmaceutical Co., Ltd. (US) 2019-11-22 CN disclosed
CN-107629059-A It can be used as the compound of ATR kinase inhibitors 沃泰克斯药物股份有限公司 2018-01-26 CN disclosed
CN-107501274-A It can be used as the compound of ATR kinase inhibitors 沃泰克斯药物股份有限公司 2017-12-22 CN disclosed
CN-107501275-A It can be used as the compound of ATR kinase inhibitors 沃泰克斯药物股份有限公司 2017-12-22 CN disclosed
CN-104903325-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2017-10-20 CN disclosed
CN-105189515-A Furopyridines as bromodomain inhibitors GLAXOSMITHKLINE IP NO 2 LTD 2015-12-23 CN disclosed
CN-105121436-A Novel pyridine derivatives HOFFMANN LA ROCHE 2015-12-02 CN disclosed