SCHEMBL28041981

SCHEMBL28041981

O=C1CCN(Cc2ccccc2)C(F)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
GAA P10253 1/20 0.41
PARP1 P09874 1/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TACR1 P25103 3/20 0.40
CYP2C19 P33261 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
TP53 P04637 1/20 0.40
MDM2 Q00987 1/20 0.40
F2 P00734 1/20 0.39
PLG P00747 1/20 0.39
ELANE P08246 1/20 0.39
CTSG P08311 1/20 0.39
CMA1 P23946 1/20 0.39
CTRC Q99895 1/20 0.39
ALDH1A1 P00352 1/20 0.38
RGS4 P49798 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24365247 0.83 PARP1 (0.46) HPGDTSHRGAAPARP1DDB1
SCHEMBL20169541 0.81 KMT2A (0.45) HPGDGAAPARP1DDB1CRBN
SCHEMBL28041842 0.81 RGS4 (0.41) HPGDTSHRGAAPARP1DDB1
SCHEMBL22873345 0.81 MAPT (0.45) SIGMAR1
SCHEMBL755504 0.81 MAPT (0.45) SIGMAR1
SCHEMBL19411417 0.80 PARP1 (0.39) HPGDTSHRGAAPARP1DDB1
SCHEMBL8924663 0.79
SCHEMBL3557054 0.79
SCHEMBL14155712 0.78 SIGMAR1 (0.42) TSHRGAASIGMAR1F2PLG
SCHEMBL14034000 0.77 PARP1 (0.39) GAAPARP1DDB1CRBNL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103288824-B Tetrahydropyridine Pyridione derivatives, its preparation method and application SHANGHAI NORMAL UNIVERSITY (CN) 2015-12-09 CN disclosed