SCHEMBL28042412

SCHEMBL28042412

Cc1cc(CC(=O)c2ccccc2)cc(C)c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.46
MAPT P10636 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
SRD5A2 P31213 2/20 0.45
KMT2A Q03164 5/20 0.44
RAB9A P51151 5/20 0.44
MEN1 O00255 4/20 0.44
NPC1 O15118 3/20 0.44
KDM4E B2RXH2 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
LMNA P02545 2/20 0.44
APAF1 O14727 1/20 0.44
MITF O75030 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
CYP3A4 P08684 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
CES1 P23141 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28042191 0.83 MAPT (0.46) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL1555065 0.81 KMT2A (0.54) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL7928075 0.80 KMT2A (0.53) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL11289129 0.79 MAPT (0.54) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL165944 0.77 CTBP2 (0.57) MAPTL3MBTL1SRD5A2KMT2ARAB9A
SCHEMBL30486043 0.77 MAPT (0.51) PLAUMAPTL3MBTL1SRD5A2KMT2A
Methyl Alcohol SCHEMBL11602292 0.75 MAPT (0.68) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL7199268 0.75 MAPT (0.67) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL24800 0.75 MAPT (0.73) PLAUMAPTL3MBTL1SRD5A2KMT2A
SCHEMBL6390145 0.74 ALDH1A1 (0.56) MAPTL3MBTL1SRD5A2KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017254-A 4-(4-((9H-purine-6-base)sulphur)phenyl)thiazolyl-2-amine derivative and preparation method and application thereof UNIV SICHUAN 2015-11-04 CN disclosed