SCHEMBL28042885

SCHEMBL28042885

CNc1cc(-c2ccc(OC(F)(F)F)cc2)nc(N2CCCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GALR2 O43603 4/20 0.51
MAPT P10636 2/20 0.48
TP53 P04637 2/20 0.48
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MCHR1 Q99705 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
ACP1 P24666 2/20 0.42
KMT2A Q03164 1/20 0.40
CCR6 P51684 2/20 0.40
CHRNA7 P36544 1/20 0.40
ABL1 P00519 1/20 0.39
BCR P11274 1/20 0.39
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.39
ALOX5 P09917 1/20 0.39
BRD4 O60885 1/20 0.39
GALR1 P47211 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043071 0.90 ABL1 (0.52) GALR2MAPTKDM4EHSD17B10MCHR1
SCHEMBL28824391 0.84 LMNA (0.46) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL21434101 0.81 KMT2A (0.61) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL16014446 0.79 GALR2 (0.46) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL21434184 0.79 GALR2 (0.53) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL21434158 0.78 TP53 (0.48) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL3997867 0.77 L3MBTL1 (0.50) GALR2KDM4EMCHR1KMT2ACHRNA7
SCHEMBL28185039 0.77 MAPT (0.48) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL4358367 0.76 KDM4E (0.50) GALR2MAPTTP53KDM4EALDH1A1
SCHEMBL4358482 0.76 ABL1 (0.58) GALR2MAPTTP53KDM4EMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143188-A Novel sulfonamide trpa1 receptor antagonists PHARMESTE S R L IN LIQUIDATION 2015-12-09 CN disclosed