SCHEMBL28043733

SCHEMBL28043733

CNc1cnn(-c2ccccc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.49
ADORA2A P29274 2/20 0.47
ADORA1 P30542 2/20 0.47
ELOVL1 Q9BW60 1/20 0.47
LSS P48449 1/20 0.42
KDM4E B2RXH2 6/20 0.42
HPGD P15428 3/20 0.42
HSD17B10 Q99714 2/20 0.41
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTT P42858 1/20 0.38
HDAC1 Q13547 1/20 0.36
MAPT P10636 2/20 0.36
NPY5R Q15761 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
NCF1 P14598 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374338 0.80 ADORA2A (0.39) P2RX7ADORA2AADORA1ELOVL1HSD17B10
SCHEMBL458507 0.74 P2RX7 (0.53) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL9468809 0.71 P2RX7 (0.55) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL6464483 0.70 HDAC1 (0.55) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL18039129 0.69 P2RX7 (0.53) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL1037429 0.69 P2RX7 (0.53) P2RX7ELOVL1LSSKDM4EHPGD
SCHEMBL11605633 0.69 P2RX7 (0.58) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL16797793 0.69 P2RX7 (0.49) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL12146363 0.69 P2RX7 (0.68) P2RX7ADORA2AADORA1ELOVL1LSS
SCHEMBL11915913 0.69 P2RX7 (0.49) P2RX7ADORA2AADORA1ELOVL1LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed