SCHEMBL28043763

SCHEMBL28043763

CCNc1cc(-c2cccc(Cl)c2CN)nc(N)n1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 3/20 0.54
HRH4 Q9H3N8 5/20 0.44
HRH3 Q9Y5N1 1/20 0.44
AURKA O14965 1/20 0.43
PDPK1 O15530 1/20 0.43
TGFBR1 P36897 1/20 0.43
AURKB Q96GD4 1/20 0.43
AGPAT2 O15120 7/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
TLR8 Q9NR97 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043809 0.87 NUDT1 (0.71) NUDT1HRH4HRH3AURKAPDPK1
SCHEMBL17315298 0.86 NUDT1 (0.73) NUDT1HRH4HRH3AURKAPDPK1
SCHEMBL15757008 0.85 NUDT1 (0.56) NUDT1HRH4HRH3AURKAPDPK1
SCHEMBL28267202 0.84 NUDT1 (0.53) NUDT1HRH4HRH3AURKAPDPK1
SCHEMBL28043914 0.80 HSP90AA1 (0.67) NUDT1HSP90AA1HSP90AB1
SCHEMBL17413783 0.80 NUDT1 (0.56) NUDT1HRH4AURKAPDPK1TGFBR1
SCHEMBL28043730 0.79 NUDT1 (0.53) NUDT1HRH4AGPAT2HSP90AA1HSP90AB1
SCHEMBL28267599 0.79 NUDT1 (0.48) NUDT1HRH4HRH3AGPAT2HSP90AA1
SCHEMBL28043729 0.79 NUDT1 (0.53) NUDT1HRH4AGPAT2HSP90AA1HSP90AB1
SCHEMBL28267166 0.77 CA1 (0.49) NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed