SCHEMBL28043809

SCHEMBL28043809

CNc1cc(-c2cccc(Cl)c2CN)nc(N)n1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 7/20 0.71
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
PTPN1 P18031 3/20 0.43
AGPAT2 O15120 5/20 0.42
HRH4 Q9H3N8 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
AURKA O14965 1/20 0.39
PDPK1 O15530 1/20 0.39
TGFBR1 P36897 1/20 0.39
ROCK1 Q13464 1/20 0.39
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043763 0.87 NUDT1 (0.54) NUDT1HSP90AA1HSP90AB1AGPAT2HRH4
SCHEMBL28267202 0.86 NUDT1 (0.53) NUDT1HSP90AA1HSP90AB1AGPAT2HRH4
SCHEMBL15757374 0.83 NUDT1 (1.00) NUDT1HSP90AA1HSP90AB1PTPN1AGPAT2
SCHEMBL29417852 0.83 NUDT1 (1.00) NUDT1HSP90AA1HSP90AB1PTPN1AGPAT2
SCHEMBL15757710 0.83 NUDT1 (0.78) NUDT1HSP90AA1HSP90AB1PTPN1AGPAT2
SCHEMBL28043746 0.83 NUDT1 (0.73) NUDT1HSP90AA1HSP90AB1PTPN1AGPAT2
SCHEMBL15757415 0.82 NUDT1 (0.77) NUDT1HSP90AA1HSP90AB1PTPN1AGPAT2
SCHEMBL28043914 0.82 HSP90AA1 (0.67) NUDT1HSP90AA1HSP90AB1ROCK1
SCHEMBL28043729 0.81 NUDT1 (0.53) NUDT1HSP90AA1HSP90AB1AGPAT2HRH4
SCHEMBL28043730 0.81 NUDT1 (0.53) NUDT1HSP90AA1HSP90AB1AGPAT2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed