SCHEMBL28044305

SCHEMBL28044305

Cc1ccc2cc(C(=O)OC(C)P(=O)(O)O)oc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.45
TAS1R3 Q7RTX0 3/20 0.41
TAS1R1 Q7RTX1 3/20 0.41
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
POLB P06746 3/20 0.39
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 2/20 0.39
HPGD P15428 3/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
AKR1B1 P15121 1/20 0.38
THRB P10828 1/20 0.37
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.37
TP53 P04637 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28044304 0.85 CYP2D6 (0.51) MAPTTAS1R3TAS1R1NPC1RAB9A
SCHEMBL28044384 0.85 NPC1 (0.39) MAPTNPC1RAB9APOLBKDM4E
SCHEMBL28044307 0.80 TAS1R3 (0.39) MAPTTAS1R3TAS1R1NPC1RAB9A
SCHEMBL10955059 0.77 MAPT (0.54) MAPTNPC1RAB9APOLBKDM4E
SCHEMBL28044297 0.77 TAS1R3 (0.59) MAPTTAS1R3TAS1R1KDM4EHPGD
SCHEMBL28044279 0.77 THRA (0.46) TAS1R3TAS1R1NPC1RAB9AKDM4E
SCHEMBL2246104 0.75 MAPT (0.51) MAPTTAS1R3TAS1R1NPC1RAB9A
SCHEMBL13155417 0.72 ALDH1A1 (0.54) MAPTTAS1R3TAS1R1NPC1RAB9A
SCHEMBL5599845 0.72 PIM1 (0.54) MAPTNPC1RAB9APOLBKDM4E
SCHEMBL11744545 0.70 NPC1 (0.47) MAPTTAS1R3TAS1R1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103130705-B Benzo five-membered unsaturated heterocycle compound or its pharmaceutical salts and preparation method thereof, pharmaceutical composition and application thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-04-20 CN claimed
CN-103130705-B Benzo five-membered unsaturated heterocycle compound or its pharmaceutical salts and preparation method thereof, pharmaceutical composition and application thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-04-20 CN disclosed