SCHEMBL28044489

SCHEMBL28044489

O=COCc1ncc(OCC(F)(F)F)c(-c2ccc(Cl)c(Cl)c2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
KIF20B Q96Q89 1/20 0.36
SLC6A3 Q01959 1/20 0.34
GRM2 Q14416 1/20 0.33
KMO O15229 2/20 0.32
CNR2 P34972 2/20 0.32
PTGES O14684 3/20 0.32
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31
TTR P02766 1/20 0.31
LMNA P02545 1/20 0.31
CRHBP P24387 1/20 0.31
MC4R P32245 1/20 0.31
CRHR2 Q13324 1/20 0.31
MPL P40238 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412314 0.80 KIF20B (0.42) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL411963 0.76 KMO (0.47) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL411960 0.74 SLC6A3 (0.41) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL31267238 0.74 MEN1 (0.40) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL21634939 0.74 MEN1 (0.40) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL28912077 0.72 GRM2 (0.44) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL21634717 0.70 TTR (0.47) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL31267253 0.70 TTR (0.47) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL21634704 0.68 NOTUM (0.46) KMT2ANPSR1MEN1MAPTHTT
SCHEMBL27924528 0.68 CNR1 (0.34) KMT2AMEN1MAPTCNR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103118680-B Heteroaryl carboxamides HOFFMAN-LA ROCHE LTD. (CH) 2015-12-16 CN disclosed