SCHEMBL28044502

SCHEMBL28044502

CCOC(=O)Cn1ncc2c1CC1CN(C(=O)OC(C)(C)C)CC21

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 8/20 0.39
NR1H2 P55055 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
GPR119 Q8TDV5 1/20 0.37
USP30 Q70CQ3 1/20 0.36
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SPR P35270 1/20 0.35
LIPE Q05469 2/20 0.35
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28044586 0.83 NR1H2 (0.44) PIK3CDNR1H2GPR119USP30SPR
SCHEMBL7989746 0.76 SMN1; SMN2 (0.39) SMN1; SMN2GPR119LMNAMEN1ALDH1A1
SCHEMBL7975140 0.74 ESR2 (0.44) NR1H2SMN1; SMN2GPR119LMNAMEN1
SCHEMBL22629402 0.72 NR1H2 (0.51) NR1H2SMN1; SMN2GPR119ALDH1A1
SCHEMBL7986449 0.70 SMN1; SMN2 (0.40) SMN1; SMN2LMNAMEN1ALDH1A1KMT2A
SCHEMBL28044510 0.68 USP30 (0.42) PIK3CDNR1H2GPR119USP30LIPE
SCHEMBL19816595 0.68 NR1H2 (0.44) NR1H2GPR119MEN1ALDH1A1KMT2A
SCHEMBL31364874 0.68 NR1H2 (0.44) NR1H2GPR119MEN1ALDH1A1KMT2A
SCHEMBL13744392 0.68 NR1H2 (0.44) NR1H2SMN1; SMN2GPR119MEN1ALDH1A1
Hydrochloric Acid SCHEMBL7989639 0.67 SMN1; SMN2 (0.39) SMN1; SMN2LMNAMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085530-A Fused tricyclic substituted amino six-membered ring derivative and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2015-11-25 CN disclosed