Quinoline

Quinoline

SCHEMBL28044618

CCc1ccc2cc[nH]c2c1.c1ccc2ncccc2c1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 2/20 0.42
CYP2A6 P11509 1/20 0.42
BACE1 P56817 4/20 0.41
NR4A2 P43354 1/20 0.40
CYP3A4 P08684 1/20 0.39
TRPA1 O75762 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
AHR P35869 1/20 0.39
ADK P55263 1/20 0.39
AXL P30530 1/20 0.38
NUDT1 P36639 1/20 0.38
PDE10A Q9Y233 1/20 0.37
KIF11 P52732 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27725634 0.89 ALDH1A1 (0.46) ALDH1A1CYP1A2CYP2A6TRPA1CA1
SCHEMBL31271 0.81 AHR (0.50) ALDH1A1CYP1A2CYP2A6BACE1AHR
Quinoline SCHEMBL27593158 0.80 CYP1A2 (0.59) ALDH1A1CYP1A2CYP2A6NR4A2CYP3A4
Quinoline SCHEMBL28292512 0.79 ALDH1A1 (0.63) ALDH1A1CYP1A2NR4A2CYP3A4TRPA1
Quinoline SCHEMBL28073739 0.79 ALDH1A1 (0.63) ALDH1A1CYP1A2NR4A2CYP3A4TRPA1
Quinoline SCHEMBL843861 0.79 ALDH1A1 (0.63) ALDH1A1CYP1A2NR4A2CYP3A4TRPA1
Quinoline SCHEMBL28816675 0.79 ALDH1A1 (0.63) ALDH1A1CYP1A2NR4A2CYP3A4TRPA1
Quinoline SCHEMBL28826923 0.79 NR4A2 (0.63) ALDH1A1CYP1A2CYP2A6NR4A2TRPA1
Quinoline SCHEMBL28046361 0.79 AHR (0.62) ALDH1A1CYP1A2CYP2A6NR4A2TRPA1
Quinoline SCHEMBL27735425 0.79 ALDH1A1 (0.54) ALDH1A1CYP1A2BACE1NR4A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073730-B monocyclic pyridine derivatives 卫材R&D管理有限公司 2017-10-13 CN disclosed
CN-105073730-A monocyclic pyridine derivatives WEI CAIR 2015-11-18 CN disclosed