SCHEMBL28044803

SCHEMBL28044803

NCc1ccc(-c2ccc3ccncc3c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 1/20 0.67
CYP2A6 P11509 1/20 0.54
MELK Q14680 1/20 0.53
HRH3 Q9Y5N1 1/20 0.48
IKBKB O14920 1/20 0.47
CHUK O15111 1/20 0.47
LCK P06239 1/20 0.47
ROCK1 Q13464 1/20 0.47
CYP19A1 P11511 3/20 0.45
TBXAS1 P24557 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.45
PIK3CD O00329 1/20 0.44
PIK3CB P42338 1/20 0.44
PIK3CG P48736 1/20 0.44
CYP17A1 P05093 4/20 0.44
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
CYP3A4 P08684 2/20 0.44
AKT1 P31749 1/20 0.43
TAAR1 Q96RJ0 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779124 0.85 MELK (0.55) PRKCZCYP2A6MELKIKBKBCHUK
SCHEMBL20031924 0.83 PRKCZ (0.62) PRKCZCYP2A6MELKCYP19A1TBXAS1
SCHEMBL29650645 0.81 PRKCZ (0.75) PRKCZROCK1CYP19A1PIK3CDPIK3CB
SCHEMBL3322974 0.81 PRKCZ (0.75) PRKCZROCK1CYP19A1PIK3CDPIK3CB
SCHEMBL18713801 0.80 PRKCZ (0.58) PRKCZMELKCYP19A1TBXAS1PIK3CD
SCHEMBL5007325 0.78 PRKCZ (0.70) PRKCZCYP19A1PIK3CDPIK3CBPIK3CG
SCHEMBL5801109 0.78 CYP19A1 (0.54) PRKCZCYP2A6MELKIKBKBCHUK
SCHEMBL31472893 0.78 CYP19A1 (0.54) PRKCZCYP2A6MELKIKBKBCHUK
SCHEMBL23555378 0.77 PRKCZ (0.68) PRKCZMELKLCKCYP19A1PIK3CD
SCHEMBL8338092 0.77 PRKCZ (0.68) PRKCZMELKLCKCYP19A1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105541713-B Isoquinoline compound and synthetic method thereof 湖南科技大学 2018-04-06 CN disclosed
CN-105541713-A Isoquinoline compound and synthetic method thereof UNIV HUNAN SCI & TECHNOLOGY 2016-05-04 CN disclosed
CN-105503722-A Method for synthesizing isoquinoline compound UNIV HUNAN SCI & TECHNOLOGY 2016-04-20 CN disclosed