SCHEMBL20031924

SCHEMBL20031924

CCc1ccc(-c2ccc3ccncc3c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 1/20 0.62
CYP17A1 P05093 3/20 0.45
CYP19A1 P11511 3/20 0.45
TBXAS1 P24557 1/20 0.45
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
CYP3A4 P08684 1/20 0.44
PIK3CD O00329 3/20 0.43
PIK3CB P42338 3/20 0.43
PIK3CG P48736 3/20 0.43
PIK3CA P42336 2/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PRKCI P41743 1/20 0.42
TDO2 P48775 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18713801 0.87 PRKCZ (0.58) PRKCZCYP17A1CYP19A1TBXAS1CYP11B1
SCHEMBL26556456 0.86 RAB9A (0.53) PRKCZCYP17A1CYP19A1CYP11B1CYP11B2
SCHEMBL26553186 0.86 RAB9A (0.53) PRKCZCYP17A1CYP19A1CYP11B1CYP11B2
SCHEMBL6114863 0.85 CYP1A2 (0.55) PRKCZCYP19A1TBXAS1ALDH1A1MAPT
SCHEMBL28044803 0.83 PRKCZ (0.67) PRKCZCYP17A1CYP19A1TBXAS1CYP11B1
SCHEMBL26556365 0.82 CYP11B2 (0.63) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL26553137 0.82 CYP11B2 (0.63) CYP17A1CYP19A1CYP11B1CYP11B2CYP3A4
SCHEMBL29650645 0.81 PRKCZ (0.75) PRKCZCYP17A1CYP19A1CYP11B1CYP11B2
SCHEMBL3322974 0.81 PRKCZ (0.75) PRKCZCYP17A1CYP19A1CYP11B1CYP11B2
SCHEMBL22826623 0.81 PRKCZ (0.44) PRKCZCYP19A1TBXAS1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018060949-A1 TRYPTOPHAN HYDROXYLASE INHIBITORS FOR USE IN THE TREATMENT OF LIVER DISEASES ROIVANT SCIENCES GMBH (CH) 2018-04-05 WO disclosed