SCHEMBL28045695

SCHEMBL28045695

O=COC(Cc1ccccc1)Cc1nnn[nH]1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
EPHX1 P07099 1/20 0.34
CYP1A2 P05177 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
CPA3 P15088 1/20 0.30
FOLH1 Q04609 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18085416 0.80 EPHX1 (0.48) CTSKCTSLCTSBEPHX1CYP1A2
SCHEMBL28814855 0.72 MMP2 (0.37) CTSKCTSLCTSBMEN1KMT2A
SCHEMBL12630161 0.69 ACE (0.44) CTSKCTSLCTSBEPHX1CYP1A2
SCHEMBL10487993 0.68 CTSK (0.41) CTSKCTSLCTSBEPHX1CYP1A2
SCHEMBL232998 0.68 NR1H2 (0.46) KMT2ATAAR1
SCHEMBL4715479 0.67 DAO (0.47) TAAR1
SCHEMBL9978690 0.67 NR1H2 (0.44) KMT2ATAAR1
SCHEMBL11395945 0.67 MDM2 (0.37) CYP1A2
SCHEMBL11528941 0.67 CYP1A2 (0.42) EPHX1CYP1A2TAAR1CPA3FOLH1
SCHEMBL5173931 0.67 NR1H2 (0.44) KMT2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121432-A Heterocyclic amides as kinase inhibitors GLAXOSMITHKLINE IP DEV LTD 2015-12-02 CN disclosed