SCHEMBL28045709

SCHEMBL28045709

CCC(=O)Nc1ccccc1C(=O)NCCc1cccc(C(C)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.48
KMT2A Q03164 1/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPC1 O15118 6/20 0.47
ITGA4 P13612 1/20 0.46
ITGB7 P26010 1/20 0.46
LMNA P02545 1/20 0.46
KDM4E B2RXH2 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MT-CO2 P00403 1/20 0.45
HDAC3 O15379 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28045659 0.87 SPR (0.53) RAB9AMTNR1AMTNR1BCYP1A2CYP3A4
SCHEMBL6097905 0.85 MT-CO2 (0.59) RAB9AKMT2ANPC1LMNAKDM4E
SCHEMBL5750887 0.75 BACE1 (0.63) RAB9AKMT2ANPC1LMNAKDM4E
SCHEMBL6098448 0.75 KDM4E (0.67) RAB9AKMT2ACYP3A4CYP2C9CYP2C19
SCHEMBL5189053 0.72 ALDH1A1 (0.62) RAB9AKMT2ANPC1LMNAKDM4E
SCHEMBL17554025 0.72 KCNH2 (0.62) RAB9AKMT2ANPC1ITGA4ITGB7
SCHEMBL28045735 0.70 MEN1 (0.69) RAB9AKMT2ANPC1
SCHEMBL29490827 0.70 MT-CO2 (0.59) RAB9ACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL22745917 0.70 MT-CO2 (0.59) RAB9ACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1826506 0.70 TAAR1 (0.54) KMT2ACYP1A2LMNAKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105198786-B Amides compound of aryl substitution and preparation method thereof, the pharmaceutical composition comprising it and its application 中国医学科学院医药生物技术研究所 2018-06-29 CN claimed
CN-105198786-A Aryl-substituted amide compound, preparing method thereof, medicine composition comprising same, and application thereof INST MED BIOTECHNOLOGY CAMS 2015-12-30 CN claimed
CN-105198786-B Amides compound of aryl substitution and preparation method thereof, the pharmaceutical composition comprising it and its application 中国医学科学院医药生物技术研究所 2018-06-29 CN disclosed
CN-105198786-A Aryl-substituted amide compound, preparing method thereof, medicine composition comprising same, and application thereof INST MED BIOTECHNOLOGY CAMS 2015-12-30 CN disclosed