SCHEMBL28045798

SCHEMBL28045798

Br[Zn]Br.[CH2]c1cnc(OC(F)F)c(-c2cccc(Cl)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 6/20 0.40
TDO2 P48775 1/20 0.38
DHFR P00374 1/20 0.37
PDE4B Q07343 1/20 0.36
ADORA1 P30542 2/20 0.35
ADORA2A P29274 1/20 0.35
CTSA P10619 2/20 0.33
KCNA5 P22460 1/20 0.33
CHEK1 O14757 1/20 0.33
LIMK1 P53667 1/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPY5R Q15761 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16043810 0.81 TDO2 (0.39) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL16045314 0.80 PDE4B (0.43) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL28045843 0.79 TDO2 (0.37) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL28604063 0.79 PDE4B (0.44) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL28045842 0.78 PDE4B (0.42) NUDT1TDO2DHFRPDE4BADORA1
Bromide SCHEMBL16044409 0.78 PDE4B (0.43) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL16045864 0.78 DRD1 (0.42) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL16047136 0.77 KCNA5 (0.39) NUDT1TDO2DHFRPDE4BADORA1
Bromide SCHEMBL16044408 0.77 PDE4B (0.43) NUDT1TDO2DHFRPDE4BADORA1
SCHEMBL16113533 0.76 PTGS2 (0.41) NUDT1TDO2DHFRADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143207-A Substituted pyridine and substituted pyrazine compounds as PDE4 inhibitors DART NEUROSCIENCE LLC 2015-12-09 CN disclosed