SCHEMBL28045843

SCHEMBL28045843

CC(Br)c1cnc(OC(F)F)c(-c2cccc(Cl)c2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.37
DHFR P00374 1/20 0.36
NUDT1 P36639 2/20 0.36
PDE4B Q07343 1/20 0.36
LIMK1 P53667 1/20 0.36
CTSA P10619 2/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KCNA5 P22460 2/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
FYN P06241 1/20 0.33
PLK1 P53350 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
PTPN11 Q06124 1/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16043810 0.90 TDO2 (0.39) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL16047136 0.88 KCNA5 (0.39) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL28045775 0.86 CTSA (0.45) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL16045405 0.80 HCRTR1 (0.35) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL28045798 0.79 NUDT1 (0.40) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL16045314 0.79 PDE4B (0.43) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL28604063 0.78 PDE4B (0.44) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL28045842 0.77 PDE4B (0.42) TDO2DHFRNUDT1PDE4BLIMK1
SCHEMBL16045864 0.77 DRD1 (0.42) TDO2DHFRNUDT1PDE4BLIMK1
Bromide SCHEMBL16044409 0.77 PDE4B (0.43) TDO2DHFRNUDT1PDE4BLIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143207-A Substituted pyridine and substituted pyrazine compounds as PDE4 inhibitors DART NEUROSCIENCE LLC 2015-12-09 CN disclosed