SCHEMBL28045824

SCHEMBL28045824

Cc1cc(-n2cncn2)c(C)cc1-n1cncn1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 3/20 0.41
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP2A6 P11509 1/20 0.38
POLB P06746 2/20 0.37
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
CYP2D6 P10635 2/20 0.36
LMNA P02545 1/20 0.36
S1PR3 Q99500 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16944266 0.82 POLB (0.42) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL26031153 0.79 CYP3A4 (0.47) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL13647554 0.77 ALDH1A1 (0.39) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL26031157 0.77 MAOB (0.48) CYP2C9CYP1A2CYP2C19CYP3A4ALDH1A1
SCHEMBL28030309 0.75 CYP19A1 (0.43) CYP2C9CYP1A2CYP2C19CYP3A4ADORA2A
SCHEMBL18394604 0.74 MYC (0.54) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL25541370 0.73 GRM7 (0.44) CYP2C9CYP1A2CYP2C19CYP3A4POLB
Cyanide SCHEMBL27958675 0.73 SMN1; SMN2 (0.41) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL1610077 0.73 KDM4E (0.41) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E
SCHEMBL1613624 0.71 S1PR3 (0.47) CYP2C9CYP1A2CYP2C19CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 148 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106243131-A 1,4 dimethyl 2,5 2 1H 1,2,4 couples triazole copper nitrate two dimension complex monocrystal and application 天津师范大学 2016-12-21 CN claimed
CN-105859750-A 1,4-dimethyl-2,5-bis-1H-double-triazole pyromellitic acid copper complex single crystal and application thereof 天津师范大学 2016-08-17 CN claimed
CN-105859755-A 1,4-dimethyl-2,5-di-1H-1,2,4-bis (triazol 1 yl) isophthalic acid cadmium complex single crystal and application 天津师范大学 2016-08-17 CN claimed
CN-105859753-A 1,4-dimethyl-2,5-di-1H-1,2,4-bis (triazol 1 yl) three-dimensional zinc complex single crystal and application 天津师范大学 2016-08-17 CN claimed
CN-105859751-A 1,4-dimethyl-2,5-di-1H-1,2,4-bis (triazol 1 yl) terephthalic acid copper complex single crystal and application 天津师范大学 2016-08-17 CN claimed
CN-105859754-A 1,4-dimethyl-2,5-bis-1H-1,2,4-double-triazole zinc mixed complex single crystal and application thereof 天津师范大学 2016-08-17 CN claimed
CN-105859786-A 1,4-dimethyl-2,5-di-1H-1,2,4-bis (triazol 1 yl) 5-methylisophthalic acid manganese complex single crystal and application 天津师范大学 2016-08-17 CN claimed
CN-105859756-A 1,4-dimethyl-2,5-di-1H-1,2,4-bis (triazol 1 yl) cadmium mixed-ligand complex single crystal and application 天津师范大学 2016-08-17 CN claimed
CN-105837603-A 1,4-dimethyl-2,5-di-1H-1,2,4-bistriazolylbiphenyldicarboxylic acid copper complex monocrystal and application thereof 天津师范大学 2016-08-10 CN claimed
CN-105837605-A 1, 4-dimethyl-2, 5-bi-1H-1, 2, 4-bis (triazol 1 yl) two-dimensional copper complex single crystal and application 天津师范大学 2016-08-10 CN claimed
CN-105503914-A Triazole isophthalic acid cadmium complex single crystal and preparation method and application thereof UNIV TIANJIN 2016-04-20 CN claimed
CN-105503910-A 1, 4-dimethyl-2, 5-dimethylene bis triazole two-dimensional zinc m-phthalate complex single crystal and application UNIV TIANJIN 2016-04-20 CN claimed
CN-105503913-A 1, 4-dimethyl-2, 5-dimethylene bis triazole cadmium terephthalate complex single crystal and application UNIV TIANJIN 2016-04-20 CN claimed
CN-105418688-A 1,4-dimethyl-2,5-dimethylene bis triazol three-dimensional nickel complex single crystal and application UNIV TIANJIN 2016-03-23 CN claimed
CN-105418657-A 1,4-dimethyl-2,5-dimethylene bis(triazole)isophthalic acid-included dimethylacetamide cadimium complex single crystal and application UNIV TIANJIN 2016-03-23 CN claimed
CN-105418660-A 1,4-dimethyl-2,5-dimethylene bis(triazole)cadimium complex single crystal and application UNIV TIANJIN 2016-03-23 CN claimed
CN-105418654-A 1,4-dimethyl-2,5-dimethylene bis(triazole) 5-methyl isophthalic acid cadimium complex single crystal and application UNIV TIANJIN 2016-03-23 CN claimed
CN-105418523-A 1,4-dimethyl-2,5-dimethylene bis(triazole)terephthalic acid single crystal and application UNIV TIANJIN 2016-03-23 CN claimed
CN-105418658-A 1,4-dimethyl-2,5-dimethylene bis triazol one-dimensional cadmium complex single crystal and application UNIV TIANJIN 2016-03-23 CN claimed
CN-105418659-A 1,4-dimethyl-2,5-dimethylene bis triazol hydroxyphenylacetic isophthalic acid cadmium complex single crystal and application UNIV TIANJIN 2016-03-23 CN claimed