SCHEMBL28046348

SCHEMBL28046348

Cc1ncccc1C(=O)OCNC(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.50
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
STING1 Q86WV6 1/20 0.42
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NAMPT P43490 1/20 0.38
ATR Q13535 1/20 0.38
KCNA5 P22460 1/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
POLB P06746 1/20 0.37
IDO1 P14902 1/20 0.37
DYRK1A Q13627 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28216226 0.81 ADRB2 (0.50) HTTL3MBTL1KCNA5IDO1SMN1; SMN2
SCHEMBL2633213 0.80 P2RX7 (0.56) P2RX7CYP3A4L3MBTL1KDM4EATR
SCHEMBL6290022 0.79 TDP1 (0.50) HTTL3MBTL1KDM4EKCNA5IDO1
SCHEMBL10033962 0.78 P2RX7 (0.67) P2RX7HTTL3MBTL1KDM4EPOLB
SCHEMBL28866297 0.77 KCNA5 (0.47) HTTL3MBTL1NAMPTKCNA5POLB
SCHEMBL29571304 0.76 TSHR (0.63) P2RX7HTTL3MBTL1SMN1; SMN2NPC1
SCHEMBL109206 0.76 TSHR (0.63) P2RX7HTTL3MBTL1SMN1; SMN2NPC1
SCHEMBL27446610 0.75 ADRB2 (0.53) KDM4ENPC1ALDH1A1RAB9A
SCHEMBL29444991 0.75 P2RX7 (0.50) P2RX7KDM4EATRPOLBSMN1; SMN2
SCHEMBL28216192 0.74 P2RX7 (0.60) P2RX7CYP2C9CYP2C19HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105101970-A Beta-lactamase inhibitors VENATORX PHARMACEUTICALS INC 2015-11-25 CN disclosed