SCHEMBL28046482

SCHEMBL28046482

Nc1cc2c(Cl)nccc2cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.44
MAPT P10636 3/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
APEX1 P27695 1/20 0.38
MAPK1 P28482 1/20 0.38
PMP22 Q01453 1/20 0.38
FGFR1 P11362 1/20 0.37
SRC P12931 1/20 0.37
PIK3CD O00329 2/20 0.37
NOS3 P29474 5/20 0.36
NOS2 P35228 5/20 0.36
NOS1 P29475 4/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PARG Q86W56 1/20 0.35
MAP4K4 O95819 1/20 0.35
F12 P00748 1/20 0.34
PLAU P00749 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14627578 0.80 NOS3 (0.50) PDPK1MAPTFGFR1SRCNOS3
SCHEMBL25368878 0.78 MAPT (0.47) MAPTLMNACYP3A4APEX1MAPK1
SCHEMBL3068849 0.74 CYP3A4 (0.43) MAPTLMNACYP3A4APEX1MAPK1
SCHEMBL558996 0.73 PDPK1 (0.53) PDPK1FGFR1SRCMEN1KMT2A
SCHEMBL4000886 0.73 CASP6 (0.49) MAPTLMNACYP3A4APEX1MAPK1
SCHEMBL558479 0.73 PDPK1 (0.44) PDPK1CYP3A4FGFR1SRCPIK3CD
SCHEMBL31686325 0.73 PDPK1 (0.40) PDPK1MAPTLMNANOS3NOS2
SCHEMBL15124778 0.73 LMNA (0.44) MAPTLMNACYP3A4APEX1MAPK1
SCHEMBL30576347 0.73 LMNA (0.44) MAPTLMNACYP3A4APEX1MAPK1
SCHEMBL22589259 0.71 LMNA (0.42) MAPTLMNACYP3A4APEX1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103261167-B 6 of replacement, 6-condenses nitrogen-containing heterocycle compound and uses thereof HOFFMAN-LA ROCHE LTD. (CH) 2016-05-04 CN disclosed