SCHEMBL28047591

SCHEMBL28047591

NNC(=O)c1cc2cccccc-2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
ALDH1A1 P00352 6/20 0.52
MAPT P10636 6/20 0.52
KDM4E B2RXH2 4/20 0.52
L3MBTL1 Q9Y468 3/20 0.52
GAA P10253 2/20 0.52
BLM P54132 2/20 0.52
LMNA P02545 2/20 0.52
NSD2 O96028 1/20 0.52
ALPL P05186 1/20 0.52
POLB P06746 1/20 0.52
ALPI P09923 1/20 0.52
ALPG P10696 1/20 0.52
APEX1 P27695 1/20 0.52
HTT P42858 1/20 0.52
RECQL P46063 1/20 0.52
CASP6 P55212 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31148960 0.92 DHODH (0.55) HDAC8MEN1KMT2AALDH1A1MAPT
SCHEMBL315040 0.90 HDAC8 (0.70) HDAC8ALDH1A1KDM4EKMOERCC5
SCHEMBL28254875 0.87 ALDH1A1 (0.68) HDAC8ALDH1A1MAPTKDM4EL3MBTL1
SCHEMBL25700071 0.87 ALDH1A1 (0.68) HDAC8ALDH1A1MAPTKDM4EL3MBTL1
SCHEMBL1706875 0.83 NPC1 (0.67) HDAC8MEN1KMT2AALDH1A1MAPT
SCHEMBL20078583 0.81 CYP3A4 (0.62) HDAC8MEN1KMT2AALDH1A1MAPT
Benzoic Acid Hydrazide SCHEMBL83514 0.81 CYP3A4 (0.62) HDAC8MEN1KMT2AALDH1A1MAPT
Benzoic Acid Hydrazide SCHEMBL4515671 0.81 CYP3A4 (0.62) HDAC8MEN1KMT2AALDH1A1MAPT
Hydrochloric Acid SCHEMBL5804936 0.81 NPC1 (0.64) HDAC8MEN1KMT2AALDH1A1MAPT
SCHEMBL3793085 0.80 ALDH1A1 (0.59) HDAC8ALDH1A1MAPTKDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102333779-B Benzopyran and benzoxex PI3K inhibitor compounds and methods of use GENENTECH, INC. (US) 2015-12-09 CN disclosed