SCHEMBL28048029

SCHEMBL28048029

Nc1c(S(=O)(=O)O)c(S(=O)(=O)O)c2ccc3ccc(S(=O)(=O)O)c4ccc1c2c34

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.42
AURKB Q96GD4 1/20 0.42
TTR P02766 1/20 0.37
CYP1A2 P05177 2/20 0.36
CTRB1 P17538 1/20 0.35
ALDH1A1 P00352 4/20 0.34
HSD17B10 Q99714 3/20 0.34
MEN1 O00255 3/20 0.34
MAPT P10636 3/20 0.34
THRB P10828 3/20 0.34
HPGD P15428 3/20 0.34
RECQL P46063 3/20 0.34
BLM P54132 3/20 0.34
KMT2A Q03164 3/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
KDM4E B2RXH2 2/20 0.34
TP53 P04637 2/20 0.34
CYP3A4 P08684 2/20 0.34
ALOX15 P16050 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30349926 0.90 AURKA (0.44) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL433199 0.90 AURKA (0.44) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL6135405 0.89 AURKA (0.40) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL6687050 0.82 CTRB1 (0.43) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL10001904 0.81 AURKA (0.47) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL18315988 0.81 CTRB1 (0.42) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL18315990 0.81 CTRB1 (0.42) AURKAAURKBCYP1A2CTRB1ALDH1A1
SCHEMBL11528264 0.79 AURKA (0.46) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL6535450 0.79 AURKA (0.38) AURKAAURKBTTRCYP1A2CTRB1
SCHEMBL17121328 0.78 AURKA (0.56) AURKAAURKBTTRCYP1A2CTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121471-A Pertuzumab variants and evaluation thereof HOFFMANN LA ROCHE 2015-12-02 CN disclosed