SCHEMBL28048864

SCHEMBL28048864

O=CCCCOc1ccncc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.47
CYP3A4 P08684 2/20 0.47
LMNA P02545 5/20 0.41
NPC1 O15118 3/20 0.41
TSHR P16473 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPK1 P28482 1/20 0.41
LTA4H P09960 2/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
STAT3 P40763 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12743776 0.80 CYP2D6 (0.59) CYP2D6CYP3A4LMNANPC1TSHR
SCHEMBL96854 0.79 KCNA3 (0.62) L3MBTL1LTA4HALDH1A1TDP1KCNA3
SCHEMBL525095 0.78 CYP2D6 (0.56) CYP2D6CYP3A4LMNANPC1TSHR
SCHEMBL19043241 0.78 NQO1 (0.58) LMNANPC1TSHRL3MBTL1LTA4H
SCHEMBL4495036 0.77 CYP2D6 (0.52) CYP2D6CYP3A4LMNANPC1TSHR
SCHEMBL19043239 0.76 DRD2 (0.51) NPC1L3MBTL1SMN1; SMN2KMT2AALDH1A1
SCHEMBL8437034 0.76 DRD2 (0.58) NPC1L3MBTL1KMT2ANPSR1KDM4E
SCHEMBL21051894 0.76 DRD4 (0.50) TSHRL3MBTL1LTA4HALDH1A1KDM4E
SCHEMBL27833683 0.76 ALDH1A1 (0.39) LMNAL3MBTL1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL5540021 0.76 DRD4 (0.51) KMT2ANPSR1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189515-A Furopyridines as bromodomain inhibitors GLAXOSMITHKLINE IP NO 2 LTD 2015-12-23 CN disclosed